Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4DRU

HCV NS5B in complex with macrocyclic INDOLE INHIBITOR

Functional Information from GO Data
ChainGOidnamespacecontents
A0003723molecular_functionRNA binding
A0003968molecular_functionRNA-dependent RNA polymerase activity
A0039694biological_processviral RNA genome replication
B0003723molecular_functionRNA binding
B0003968molecular_functionRNA-dependent RNA polymerase activity
B0039694biological_processviral RNA genome replication
Functional Information from PDB Data
site_idAC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE 0LN A 601
ChainResidue
AHIS34
AVAL37
ALEU392
AALA395
AALA396
AHIS428
AVAL494
AARG503

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 602
ChainResidue
ALYS51
ACYS223
AHOH856
AARG48

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 603
ChainResidue
ALYS79
AASP244
AHOH918
BLEU68

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 604
ChainResidue
AHIS475
ASER476
AHOH834

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 605
ChainResidue
ALEU60
ALEU68
AVAL235
BLYS79
BASP244

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GOL A 606
ChainResidue
ALEU83
AILE85
ATRP123
AHOH755

site_idAC7
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL A 607
ChainResidue
AGLY8
AALA9
ALEU10
AILE11
AGLN49
AHOH850
BGLU341

site_idAC8
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 601
ChainResidue
BARG505
BVAL530
BARG531
BTHR532

site_idAC9
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 602
ChainResidue
AARG114
BPRO22
BILE23
BASN24
BALA400
BARG401
BHOH1061

site_idBC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 603
ChainResidue
BTHR287
BSER288
BASN291
BGLY317
BASP318
BHOH844
BHOH1019

site_idBC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 B 604
ChainResidue
BLYS209
BARG380
BTYR382

site_idBC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 605
ChainResidue
BARG48
BLYS51
BARG158
BCYS223
BHOH1033

site_idBC4
Number of Residues2
DetailsBINDING SITE FOR RESIDUE SO4 B 606
ChainResidue
BARG43
BHOH882

site_idBC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 B 607
ChainResidue
BLEU474
BTYR477
BSO4608

site_idBC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 608
ChainResidue
BHIS475
BSER476
BSO4607
BHOH933

site_idBC7
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 609
ChainResidue
BTRP208
BLEU360
BTYR382
BHOH731

site_idBC8
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 B 610
ChainResidue
BGLU440
BARG517
BHOH774

site_idBC9
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 611
ChainResidue
BCYS366
BSER368
BLEU384
BMET414
BTYR448

site_idCC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL B 612
ChainResidue
BGLU361
BASN369
BSER371
BSER478
BGLU481
BARG484

site_idCC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL B 613
ChainResidue
ATHR130
AGLU131
AARG254
AGLU258
BLEU127
BPRO247
BGLN251

site_idCC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL B 614
ChainResidue
BARG254
BGLU258
ALEU127
APRO247
AGLU248
BTHR130

site_idCC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL B 615
ChainResidue
AASP244
AHOH763
BARG234

site_idCC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL B 616
ChainResidue
BARG386
BTHR390
BARG394

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P26663
ChainResidueDetails
AASP220
AASP318
AASP319
BASP220
BASP318
BASP319

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: Phosphoserine; by host => ECO:0000250|UniProtKB:P26662
ChainResidueDetails
ASER29
ASER42
BSER29
BSER42

222624

PDB entries from 2024-07-17

PDB statisticsPDBj update infoContact PDBjnumon