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4DRI

Co-crystal structure of the PPIase domain of FKBP51, Rapamycin and the FRB fragment of mTOR

Functional Information from GO Data
ChainGOidnamespacecontents
A0003755molecular_functionpeptidyl-prolyl cis-trans isomerase activity
B0044877molecular_functionprotein-containing complex binding
Functional Information from PDB Data
site_idAC1
Number of Residues26
DetailsBINDING SITE FOR RESIDUE RAP A 201
ChainResidue
ATYR57
ATRP90
ATYR113
AILE122
APHE130
AHOH316
AHOH353
AHOH366
AHOH386
BLEU2031
BGLU2032
APHE67
BSER2035
BPHE2039
BTHR2098
BASP2102
BTYR2105
BPHE2108
BHOH2219
AASP68
AARG73
APHE77
AGLY84
AGLN85
AVAL86
AILE87

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N-acetylmethionine => ECO:0007744|PubMed:19413330
ChainResidueDetails
AMET1

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER13

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0000269|PubMed:28147277
ChainResidueDetails
ALYS28

223532

PDB entries from 2024-08-07

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