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4CLB

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH IBET-295

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1169
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135
AHOH2179
AHOH2280

site_idAC2
Number of Residues11
DetailsBINDING SITE FOR RESIDUE 83T A 1170
ChainResidue
ALEU92
ALEU94
AASN140
AILE146
AMET149
ALYS155
AHOH2171
AHOH2282
AHOH2283
AGLN59
ATRP81

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

219140

PDB entries from 2024-05-01

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