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4CL9

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH I-BET295

Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1169
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135

site_idAC2
Number of Residues17
DetailsBINDING SITE FOR RESIDUE IES A 1170
ChainResidue
ALYS91
AASN93
ALEU94
AASP96
AASN140
AASP145
AILE146
AHOH2114
AHOH2128
AHOH2145
AHOH2228
AHOH2229
AHOH2231
ATRP81
APRO82
AGLN84
AGLN85

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

222926

PDB entries from 2024-07-24

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