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4CI4

Structural basis for GL479 a dual Peroxisome Proliferator-Activated Receptor alpha agonist

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE Y1N A 1468
ChainResidue
APHE273
AMET355
AHIS440
AVAL444
ALEU460
ATYR464
ACYS276
AGLN277
ATHR279
ASER280
ATYR314
APHE318
ALEU321
AVAL332

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues129
DetailsRegion: {"description":"Required for heterodimerization with RXRA"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues3
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"19116277","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"3ET1","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues1
DetailsSite: {"description":"Essential for heterodimerization with RXRA"}
ChainResidueDetails

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PDB entries from 2025-12-17

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