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4CGO

Leishmania major N-myristoyltransferase in complex with a thienopyrimidine inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004379molecular_functionglycylpeptide N-tetradecanoyltransferase activity
A0005829cellular_componentcytosol
A0006499biological_processN-terminal protein myristoylation
A0016740molecular_functiontransferase activity
A0016746molecular_functionacyltransferase activity
A0046872molecular_functionmetal ion binding
A0072657biological_processprotein localization to membrane
Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE MG A 1000
ChainResidue
ALEU175
AGLU177
ALYS178
AARG179
ALEU180
AMYA1001

site_idAC2
Number of Residues36
DetailsBINDING SITE FOR RESIDUE MYA A 1001
ChainResidue
ATRP15
AASN79
ATYR80
AVAL81
APHE168
ALEU169
ACYS170
AVAL171
AARG176
AGLU177
ALYS178
AARG179
ALEU180
AALA181
APRO182
ATHR189
AVAL192
ATRP198
ATYR202
ATHR203
ALEU208
ATYR404
AMG1000
AHOH2001
AHOH2002
AHOH2345
AHOH2351
AHOH2569
AHOH2570
AHOH2571
AHOH2572
AHOH2573
AHOH2574
AHIS12
AALA13
APHE14

site_idAC3
Number of Residues13
DetailsBINDING SITE FOR RESIDUE 6KV A 1422
ChainResidue
APHE90
ATYR92
AASN167
ATHR203
AGLY205
ATYR217
AHIS219
ATYR345
AHIS398
ALEU421
A6KV1423
AHOH2190
AHOH2368

site_idAC4
Number of Residues12
DetailsBINDING SITE FOR RESIDUE 6KV A 1423
ChainResidue
AVAL81
AGLU82
AASP83
APHE88
APHE90
APHE232
ASER330
ALEU341
AALA343
AASN376
AASP396
A6KV1422

Functional Information from PROSITE/UniProt
site_idPS00975
Number of Residues9
DetailsNMT_1 Myristoyl-CoA:protein N-myristoyltransferase signature 1. EINFLCvHK
ChainResidueDetails
AGLU165-LYS173

site_idPS00976
Number of Residues7
DetailsNMT_2 Myristoyl-CoA:protein N-myristoyltransferase signature 2. KFGaGDG
ChainResidueDetails
ALYS391-GLY397

239149

数据于2025-07-23公开中

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