4CGO
Leishmania major N-myristoyltransferase in complex with a thienopyrimidine inhibitor
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0004379 | molecular_function | glycylpeptide N-tetradecanoyltransferase activity |
A | 0005829 | cellular_component | cytosol |
A | 0006499 | biological_process | N-terminal protein myristoylation |
A | 0016740 | molecular_function | transferase activity |
A | 0016746 | molecular_function | acyltransferase activity |
A | 0046872 | molecular_function | metal ion binding |
A | 0072657 | biological_process | protein localization to membrane |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE MG A 1000 |
Chain | Residue |
A | LEU175 |
A | GLU177 |
A | LYS178 |
A | ARG179 |
A | LEU180 |
A | MYA1001 |
site_id | AC2 |
Number of Residues | 36 |
Details | BINDING SITE FOR RESIDUE MYA A 1001 |
Chain | Residue |
A | TRP15 |
A | ASN79 |
A | TYR80 |
A | VAL81 |
A | PHE168 |
A | LEU169 |
A | CYS170 |
A | VAL171 |
A | ARG176 |
A | GLU177 |
A | LYS178 |
A | ARG179 |
A | LEU180 |
A | ALA181 |
A | PRO182 |
A | THR189 |
A | VAL192 |
A | TRP198 |
A | TYR202 |
A | THR203 |
A | LEU208 |
A | TYR404 |
A | MG1000 |
A | HOH2001 |
A | HOH2002 |
A | HOH2345 |
A | HOH2351 |
A | HOH2569 |
A | HOH2570 |
A | HOH2571 |
A | HOH2572 |
A | HOH2573 |
A | HOH2574 |
A | HIS12 |
A | ALA13 |
A | PHE14 |
site_id | AC3 |
Number of Residues | 13 |
Details | BINDING SITE FOR RESIDUE 6KV A 1422 |
Chain | Residue |
A | PHE90 |
A | TYR92 |
A | ASN167 |
A | THR203 |
A | GLY205 |
A | TYR217 |
A | HIS219 |
A | TYR345 |
A | HIS398 |
A | LEU421 |
A | 6KV1423 |
A | HOH2190 |
A | HOH2368 |
site_id | AC4 |
Number of Residues | 12 |
Details | BINDING SITE FOR RESIDUE 6KV A 1423 |
Chain | Residue |
A | VAL81 |
A | GLU82 |
A | ASP83 |
A | PHE88 |
A | PHE90 |
A | PHE232 |
A | SER330 |
A | LEU341 |
A | ALA343 |
A | ASN376 |
A | ASP396 |
A | 6KV1422 |
Functional Information from PROSITE/UniProt