Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4CFC

Interrogating HIV integrase for compounds that bind- a SAMPL challenge

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 1210
ChainResidue
BTHR66
BHIS67
BLYS111
BLYS136
BLYS159
BHOH2033

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1210
ChainResidue
ALYS159
AHOH2005
AHOH2043
ATHR66
AHIS67
ALYS111

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 1211
ChainResidue
BLYS71
BHIS171
BLEU172
BHOH2039

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1211
ChainResidue
ALYS71
AARG166
AHIS171
ALEU172
AHOH2050

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1212
ChainResidue
AGLY94
ASER123
ATHR124
ATHR125
AHOH2020
AHOH2038

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 1212
ChainResidue
BGLY94
BSER123
BTHR124
BTHR125
BHOH2013
BHOH2014
BHOH2028

site_idAC7
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1213
ChainResidue
AGLU85
APHE100
ALYS103
BARG107

site_idAC8
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 1213
ChainResidue
AARG107
BGLU85
BPHE100
BLYS103

site_idAC9
Number of Residues6
DetailsBINDING SITE FOR RESIDUE ACT A 1214
ChainResidue
ATYR99
ALYS103
AHOH2025
AHOH2063
BACT1214
BHOH2040

site_idBC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE ACT B 1214
ChainResidue
AACT1214
AHOH2009
AHOH2011
BTYR99
BLYS103

site_idBC2
Number of Residues1
DetailsBINDING SITE FOR RESIDUE CL B 1215
ChainResidue
BHIS185

site_idBC3
Number of Residues1
DetailsBINDING SITE FOR RESIDUE CL A 1215
ChainResidue
AHIS185

site_idBC4
Number of Residues8
DetailsBINDING SITE FOR RESIDUE 7NV A 1216
ChainResidue
AASP167
AGLN168
AALA169
AGLU170
AHIS171
ATHR174
BGLN95
BALA128

site_idBC5
Number of Residues8
DetailsBINDING SITE FOR RESIDUE 7NV B 1216
ChainResidue
AGLN95
AALA128
BASP167
BGLN168
BALA169
BGLU170
BHIS171
BTHR174

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING:
ChainResidueDetails
AASP64
AASP116
BASP64
BASP116

site_idSWS_FT_FI2
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P04585
ChainResidueDetails
AGLU152
BGLU152

219140

PDB entries from 2024-05-01

PDB statisticsPDBj update infoContact PDBjnumon