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4C7I

Leismania major N-myristoyltransferase in complex with a peptidomimetic (-OH) molecule

Functional Information from GO Data
ChainGOidnamespacecontents
A0004379molecular_functionglycylpeptide N-tetradecanoyltransferase activity
A0005829cellular_componentcytosol
A0006499biological_processN-terminal protein myristoylation
A0016740molecular_functiontransferase activity
A0016746molecular_functionacyltransferase activity
A0046872molecular_functionmetal ion binding
A0072657biological_processprotein localization to membrane
Functional Information from PDB Data
site_idAC1
Number of Residues36
DetailsBINDING SITE FOR RESIDUE MYA A 1422
ChainResidue
AHIS12
AVAL171
AARG176
AGLU177
ALYS178
AARG179
ALEU180
AALA181
APRO182
ATHR189
AVAL192
AALA13
ATRP198
ATYR202
ATHR203
ALEU208
ATYR404
AMG1423
AJJ11424
AHOH2004
AHOH2328
AHOH2333
APHE14
AHOH2575
AHOH2576
AHOH2577
AHOH2578
AHOH2579
AHOH2580
AHOH2582
ATRP15
AASN79
AVAL81
APHE168
ALEU169
ACYS170

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE MG A 1423
ChainResidue
ALEU175
AGLU177
ALYS178
AARG179
ALEU180
AMYA1422

site_idAC3
Number of Residues23
DetailsBINDING SITE FOR RESIDUE JJ1 A 1424
ChainResidue
ATYR80
AASP83
AASP84
AASP85
AASN167
ATHR203
ATYR217
AHIS219
APHE232
ASER233
ATYR253
AALA394
AGLY395
AASP396
AGLY397
AMYA1422
ADMS1425
ADMS1426
AHOH2185
AHOH2189
AHOH2317
AHOH2534
AHOH2554

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE DMS A 1425
ChainResidue
APHE88
APHE90
ASER330
AJJ11424
AHOH2508

site_idAC5
Number of Residues7
DetailsBINDING SITE FOR RESIDUE DMS A 1426
ChainResidue
APHE90
ATYR92
ATYR217
ATYR345
AMET420
AJJ11424
AHOH2508

Functional Information from PROSITE/UniProt
site_idPS00975
Number of Residues9
DetailsNMT_1 Myristoyl-CoA:protein N-myristoyltransferase signature 1. EINFLCvHK
ChainResidueDetails
AGLU165-LYS173

site_idPS00976
Number of Residues7
DetailsNMT_2 Myristoyl-CoA:protein N-myristoyltransferase signature 2. KFGaGDG
ChainResidueDetails
ALYS391-GLY397

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PDB entries from 2025-06-18

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