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4C6X

Crystal structure of M. tuberculosis C171Q KasA in complex with thiolactomycin (TLM)

Functional Information from GO Data
ChainGOidnamespacecontents
A0016746molecular_functionacyltransferase activity
B0016746molecular_functionacyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1417
ChainResidue
AARG219
AASP233
AHOH2279

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE K B 1417
ChainResidue
BASN309
BALA310
BHIS311
BGLU354
BASN399
BASN400

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE K A 1418
ChainResidue
AASN309
AALA310
AHIS311
AGLU354
AASN399
AASN400

site_idAC4
Number of Residues14
DetailsBINDING SITE FOR RESIDUE TLM A 1419
ChainResidue
AGLN171
AVAL278
AALA279
APRO280
AHIS311
ATHR313
AHIS345
APHE402
AGLY403
APHE404
AGLY406
AHOH2243
AHOH2322
AHOH2438

site_idAC5
Number of Residues14
DetailsBINDING SITE FOR RESIDUE TLM B 1418
ChainResidue
BGLN171
BPHE237
BVAL278
BALA279
BPRO280
BHIS311
BTHR313
BHIS345
BPHE402
BGLY403
BPHE404
BGLY406
BHOH2264
BHOH2315

site_idAC6
Number of Residues16
DetailsBINDING SITE FOR RESIDUE M7U A 1420
ChainResidue
AGLY115
AGLU120
AALA170
AGLU199
AGLY200
APRO201
AILE202
AGLU203
ALEU205
AALA209
APHE239
AGLY240
AGLU241
AHIS345
AHOH2439
BILE145

site_idAC7
Number of Residues15
DetailsBINDING SITE FOR RESIDUE M7U B 1419
ChainResidue
AILE145
BGLY115
BGLU120
BALA170
BGLU199
BGLY200
BPRO201
BGLU203
BALA209
BPHE239
BGLY240
BHIS345
BILE347
BHOH2316
BHOH2317

site_idAC8
Number of Residues15
DetailsBINDING SITE FOR RESIDUE EPE A 1421
ChainResidue
AASP332
AGLN333
AASP381
ALEU382
AASP383
AHOH2381
AHOH2386
AHOH2401
AHOH2440
AHOH2441
AHOH2442
BARG78
BARG79
BLYS136
BHOH2163

219869

PDB entries from 2024-05-15

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