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4BVW

Identification of small molecule inhibitors selective for apo(a) kringles KIV-7, KIV-10 and KV.

Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL A 1079
ChainResidue
AHIS3
ASER8
ATYR9
AHOH2002

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL B 1079
ChainResidue
BTYR40
BPRO41
BASN42
BGLY43

site_idAC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A 1081
ChainResidue
AHKY1080
AARG35

site_idAC4
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL B 1080
ChainResidue
BTYR2
BGLN77

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO B 1081
ChainResidue
AARG20
BTYR2
BILE57
BGLN77

site_idAC6
Number of Residues8
DetailsBINDING SITE FOR RESIDUE HKY A 1080
ChainResidue
AASP54
AGLU56
ATRP60
ATYR62
AARG69
ATRP70
ACL1081
AHOH2054

site_idAC7
Number of Residues7
DetailsBINDING SITE FOR RESIDUE HKY B 1082
ChainResidue
BASP54
BGLU56
BTRP60
BTYR62
BARG69
BTRP70
BHOH2051

Functional Information from PROSITE/UniProt
site_idPS00021
Number of Residues13
DetailsKRINGLE_1 Kringle domain signature. YCRNpdaeirp.WC
ChainResidueDetails
ATYR49-CYS61

218853

PDB entries from 2024-04-24

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