Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4BU8

Crystal structure of human tankyrase 2 in complex with 4-(4-oxo-1,4- dihydroquinazolin-2-yl)benzonitrile

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
C0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 2162
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN C 2162
ChainResidue
CCYS1081
CHIS1084
CCYS1089
CCYS1092

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 C 2163
ChainResidue
CHIS979
CARG980
CLYS1067
CGLN1070
CHOH3041
CHOH3049
CARG977

site_idAC4
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 A 2163
ChainResidue
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070
AHOH3043
AHOH3051
AHOH3162

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 2164
ChainResidue
AASN990
AARG991
APRO1160
AGLU1161
AHOH3067
AHOH3070

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 C 2164
ChainResidue
CASN990
CARG991
CPRO1160
CGLU1161
CHOH3064
CHOH3067

site_idAC7
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 27F A 2165
ChainResidue
AHIS1031
AGLY1032
ASER1033
APHE1035
ATYR1050
ATYR1060
ALYS1067
ASER1068
ATYR1071
AGLU1138

site_idAC8
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 27F C 2165
ChainResidue
CHIS1031
CGLY1032
CSER1033
CPHE1035
CTYR1050
CTYR1060
CLYS1067
CSER1068
CTYR1071
CGLU1138

site_idAC9
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 2166
ChainResidue
APRO1129
ASER1130
AVAL1131
AASN1132
AGLY1133

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092
CCYS1081
CHIS1084
CCYS1089
CCYS1092

219140

PDB entries from 2024-05-01

PDB statisticsPDBj update infoContact PDBjnumon