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4BJB

Crystal structure of human tankyrase 2 in complex with PJ-34

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 A 2162
ChainResidue
AARG977
AHIS979
AARG980
ALYS1067
AASN1132
AHOH2006
AHOH2029
AHOH2079

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 2163
ChainResidue
AARG991
APRO1160
AGLU1161
AASN990

site_idAC3
Number of Residues8
DetailsBINDING SITE FOR RESIDUE GOL A 2164
ChainResidue
AARG1128
APRO1129
ASER1130
ASER1130
AVAL1131
AVAL1131
AASN1132
AASN1132

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 2165
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC5
Number of Residues9
DetailsBINDING SITE FOR RESIDUE P34 A 2166
ChainResidue
AHIS1031
AGLY1032
ATYR1060
AALA1062
ALYS1067
ASER1068
ATYR1071
AILE1075
AGLU1138

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"O95271","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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