3ZRA
Structural basis for agonism and antagonism for a set of chemically related progesterone receptor modulators
Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 12 |
| Details | BINDING SITE FOR RESIDUE ORB A 1000 |
| Chain | Residue |
| A | LEU715 |
| A | CYS891 |
| A | PHE905 |
| A | MET909 |
| A | LEU718 |
| A | ASN719 |
| A | LEU721 |
| A | MET756 |
| A | MET759 |
| A | VAL760 |
| A | LEU763 |
| A | TYR890 |
| site_id | AC2 |
| Number of Residues | 13 |
| Details | BINDING SITE FOR RESIDUE ORB B 1000 |
| Chain | Residue |
| B | LEU715 |
| B | LEU718 |
| B | ASN719 |
| B | TRP755 |
| B | MET756 |
| B | MET759 |
| B | VAL760 |
| B | MET801 |
| B | LEU887 |
| B | TYR890 |
| B | CYS891 |
| B | PHE905 |
| B | MET909 |
| site_id | AC3 |
| Number of Residues | 4 |
| Details | BINDING SITE FOR RESIDUE SO4 A 1933 |
| Chain | Residue |
| A | PRO737 |
| A | GLY738 |
| A | ARG740 |
| A | ASN741 |
Functional Information from SwissProt/UniProt
| site_id | SWS_FT_FI1 |
| Number of Residues | 2 |
| Details | Binding site: {"evidences":[{"source":"PubMed","id":"9620806","evidenceCode":"ECO:0000269"}]} |
| Chain | Residue | Details |






