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3ZRA

Structural basis for agonism and antagonism for a set of chemically related progesterone receptor modulators

Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE ORB A 1000
ChainResidue
ALEU715
ACYS891
APHE905
AMET909
ALEU718
AASN719
ALEU721
AMET756
AMET759
AVAL760
ALEU763
ATYR890

site_idAC2
Number of Residues13
DetailsBINDING SITE FOR RESIDUE ORB B 1000
ChainResidue
BLEU715
BLEU718
BASN719
BTRP755
BMET756
BMET759
BVAL760
BMET801
BLEU887
BTYR890
BCYS891
BPHE905
BMET909

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1933
ChainResidue
APRO737
AGLY738
AARG740
AASN741

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9620806","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246905

PDB entries from 2025-12-31

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