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3WZ8

Endothiapepsin in complex with Gewald reaction-derived inhibitor (8)

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues18
DetailsBINDING SITE FOR RESIDUE IXV A 401
ChainResidue
AILE10
AGLY221
ATHR222
ATHR223
ATYR226
AILE300
AILE304
AHOH669
AHOH738
AHOH1045
AASP15
AASP33
ATYR79
AGLY80
AASP81
ASER83
APHE116
AASP119

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PEG A 402
ChainResidue
APRO61
ASER62
AALA67
ALYS68
ALEU69
ATYR90

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE DMS A 403
ChainResidue
AGLY37
AILE77
ASER78
APHE194
AHOH522
AHOH748
AHOH1037

Functional Information from PROSITE/UniProt
site_idPS00141
Number of Residues12
DetailsASP_PROTEASE Eukaryotic and viral aspartyl proteases active site. LDFDTGSSDLWV
ChainResidueDetails
ALEU32-VAL43
AGLY216-LEU227

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE:
ChainResidueDetails
AASP35
ASER199

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PDB entries from 2024-07-10

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