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3W69

Crystal structure of human mdm2 with a dihydroimidazothiazole inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0043066biological_processnegative regulation of apoptotic process
A0051726biological_processregulation of cell cycle
B0005634cellular_componentnucleus
B0043066biological_processnegative regulation of apoptotic process
B0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE LTZ A 201
ChainResidue
ALEU54
BTHR26
BMET50
BLEU54
BTYR100
BTYR104
BLTZ201
AGLY58
AILE61
AGLN72
AVAL93
AHIS96
ATYR100
AHOH306
AHOH313

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 202
ChainResidue
AGLU95
AHIS96
AARG97
ALYS98
AHOH343
AHOH361
AHOH365

site_idAC3
Number of Residues16
DetailsBINDING SITE FOR RESIDUE LTZ B 201
ChainResidue
AGLU25
ALEU54
ATYR104
ALTZ201
AHOH308
AHOH310
BLEU54
BGLY58
BILE61
BGLN72
BVAL93
BHIS96
BILE99
BTYR100
BSO4203
BHOH316

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 202
ChainResidue
AARG65
BLYS94
BHIS96
BARG97
BHOH304
BHOH342

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 203
ChainResidue
BVAL93
BLYS94
BHIS96
BLTZ201

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PDB entries from 2024-07-17

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