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3W5R

Crystal structure of complexes of vitamin D receptor ligand binding domain with lithocholic acid derivatives

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE LOA A 500
ChainResidue
ATYR143
AILE306
AHIS393
AVAL414
AHOH605
AVAL230
AILE264
AILE267
ASER271
ASER274
ATRP282
AVAL296
AHIS301

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:15065852, ECO:0007744|PDB:1RK3
ChainResidueDetails
ATYR143
AMET280
ALYS317
ALEU321
AVAL348

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PDB entries from 2024-07-10

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