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3VTD

Crystal structure of rat vitamin D receptor bound to a partial agonist 26-adamantyl-23-yne-19-norvitammin D ADTK4

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE TKD A 500
ChainResidue
ATYR143
ATRP282
AVAL296
AHIS301
AHIS393
ALEU410
ALEU223
AALA227
AVAL230
ASER233
AMET268
AARG270
ASER271
ASER274

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:15065852, ECO:0007744|PDB:1RK3
ChainResidueDetails
ATYR143
AMET280
ALYS317
ALEU321
AVAL348

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PDB entries from 2024-07-17

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