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3VT6

Crystal structure of rat VDR-LBD with 2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE 5YI A 500
ChainResidue
ATYR143
ATRP282
ACYS284
AVAL296
AHIS301
AHIS393
AHOH620
APHE150
ALEU223
AVAL230
ATYR232
ASER233
AARG270
ASER271
ASER274

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:15065852, ECO:0007744|PDB:1RK3
ChainResidueDetails
ALYS317
ALEU321
AMET280
ATYR143
AVAL348

221051

PDB entries from 2024-06-12

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