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3VQE

HIV-1 IN core domain in complex with [1-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]methanol

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CD A 1001
ChainResidue
ACYS65
AHIS67
AGLU92
BASP131

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD A 1002
ChainResidue
BHOH402
ACYS65
AGLU92
AASP116
ACL1003
AHOH1106

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL A 1003
ChainResidue
ACYS65
AASP116
AASN120
ACD1002

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1004
ChainResidue
ALYS71
AARG166
AGLU170
AHIS171
ALEU172
AHOH1126

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1005
ChainResidue
ATHR66
AHIS67
ALYS159
BARG127

site_idAC6
Number of Residues8
DetailsBINDING SITE FOR RESIDUE FMQ A 1006
ChainResidue
AHIS185
AARG187
ASER195
AGLY197
AGLU198
AVAL201
BPRO109
BILE204

site_idAC7
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CD B 301
ChainResidue
AASP131
BCYS65
BHIS67
BGLU92

site_idAC8
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD B 302
ChainResidue
AHOH1105
BCYS65
BGLU92
BASP116
BCL303
BHOH403

site_idAC9
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL B 303
ChainResidue
BCYS65
BASP116
BASN120
BCD302

site_idBC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 304
ChainResidue
BLYS71
BARG166
BGLU170
BHIS171
BLEU172
BHOH419
BHOH432

site_idBC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 305
ChainResidue
AARG127
BTHR66
BHIS67
BLYS159

site_idBC3
Number of Residues10
DetailsBINDING SITE FOR RESIDUE FMQ B 306
ChainResidue
APRO109
ALYS111
AILE204
BHIS185
BARG187
BSER195
BGLY197
BGLU198
BVAL201
BHOH405

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PDB entries from 2025-06-11

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