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3VQ5

HIV-1 IN core domain in complex with N-METHYL-1-(4-METHYL-2-PHENYL-1,3-THIAZOL-5-YL)METHANAMINE

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CD A 1001
ChainResidue
ACYS65
AHIS67
AGLU92
ACD1002
BASP131

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE CD A 1002
ChainResidue
ACL1003
AHOH1103
AHOH1106
ACYS65
AGLU92
AASP116
ACD1001

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL A 1003
ChainResidue
ACYS65
AASP116
AASN120
ACD1002

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1004
ChainResidue
ALYS71
AHIS171
ALEU172
AHOH1148

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1005
ChainResidue
ATHR66
AHIS67
ALYS159
BARG127
BHOH438

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1006
ChainResidue
AGLN95
AGLY123
AALA124
ATHR125
AARG187
AHOH1108

site_idAC7
Number of Residues7
DetailsBINDING SITE FOR RESIDUE MMJ A 1007
ChainResidue
AARG107
APRO109
AILE204
AASP207
BHIS185
BGLY197
BGLU198

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CD B 301
ChainResidue
AASP131
BCYS65
BHIS67
BGLU92
BCD302

site_idAC9
Number of Residues7
DetailsBINDING SITE FOR RESIDUE CD B 302
ChainResidue
BCYS65
BGLU92
BASP116
BCD301
BCL303
BHOH403
BHOH404

site_idBC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CL B 303
ChainResidue
BCYS65
BGLU92
BASP116
BASN120
BCD302

site_idBC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 304
ChainResidue
BLYS71
BARG166
BGLU170
BHIS171
BLEU172
BHOH424

site_idBC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 305
ChainResidue
AARG127
AHOH1143
BTHR66
BHIS67
BLYS159

site_idBC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 306
ChainResidue
BGLY123
BALA124
BTHR125
BARG187
BHOH420
BHOH445

site_idBC5
Number of Residues7
DetailsBINDING SITE FOR RESIDUE MMJ B 307
ChainResidue
AHIS185
AGLY197
AGLU198
BARG107
BPRO109
BILE204
BASP207

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PDB entries from 2024-09-18

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