3V49
Structure of ar lbd with activator peptide and sarm inhibitor 1
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 17 |
Details | BINDING SITE FOR RESIDUE PK0 A 950 |
Chain | Residue |
A | LEU704 |
A | PHE764 |
A | MET780 |
A | MET787 |
A | HIS874 |
A | THR877 |
A | ILE899 |
A | VAL903 |
A | HOH2007 |
A | ASN705 |
A | GLY708 |
A | TRP741 |
A | MET742 |
A | MET745 |
A | VAL746 |
A | MET749 |
A | ARG752 |
site_id | AC2 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE SO4 A 1300 |
Chain | Residue |
A | SER696 |
A | PHE697 |
A | LYS777 |
A | SER853 |
A | HOH2073 |
site_id | AC3 |
Number of Residues | 18 |
Details | BINDING SITE FOR CHAIN B OF ANDROGEN RECEPTOR, ACTIVATOR PEPTIDE |
Chain | Residue |
A | LYS717 |
A | LYS720 |
A | ARG726 |
A | GLN733 |
A | MET734 |
A | GLN738 |
A | ARG871 |
A | MET894 |
A | GLU897 |
A | LYS912 |
A | HOH2081 |
A | HOH2181 |
B | HOH2029 |
B | HOH2107 |
B | HOH2161 |
B | HOH2165 |
B | HOH2227 |
B | HOH2228 |
Functional Information from SwissProt/UniProt
Chain | Residue | Details |
A | GLU706 |
Chain | Residue | Details |
A | SER753 | |
A | PHE878 |
site_id | SWS_FT_FI3 |
Number of Residues | 1 |
Details | SITE: Interaction with coactivator LXXL and FXXFY motifs => ECO:0000269|PubMed:25091737 |
Chain | Residue | Details |
A | ALA721 |
site_id | SWS_FT_FI4 |
Number of Residues | 1 |
Details | SITE: Interaction with coactivator FXXLF and FXXFY motifs => ECO:0000269|PubMed:25091737 |
Chain | Residue | Details |
A | ILE898 |
site_id | SWS_FT_FI5 |
Number of Residues | 1 |
Details | MOD_RES: Phosphotyrosine; by CSK => ECO:0000269|PubMed:17045208 |
Chain | Residue | Details |
A | PHE916 |
site_id | SWS_FT_FI6 |
Number of Residues | 3 |
Details | CROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:19345326 |
Chain | Residue | Details |
A | ARG846 | |
A | ASN848 |