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3UWI

Bovine trypsin variant X(tripleGlu217Phe227) in complex with small molecule inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004175molecular_functionendopeptidase activity
A0004252molecular_functionserine-type endopeptidase activity
A0005515molecular_functionprotein binding
A0005576cellular_componentextracellular region
A0005615cellular_componentextracellular space
A0006508biological_processproteolysis
A0007586biological_processdigestion
A0008236molecular_functionserine-type peptidase activity
A0046872molecular_functionmetal ion binding
A0097180cellular_componentserine protease inhibitor complex
A0097655molecular_functionserpin family protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA A 480
ChainResidue
AGLU70
AASN72
AVAL75
AGLU80
AHOH1010
AHOH1083

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE SO4 A 481
ChainResidue
ASER195
AANH487
AHOH1109
AHOH1174
AHOH1177
AHOH1185
AHOH1260
AHIS57
AGLN192
AGLY193

site_idAC3
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 A 482
ChainResidue
APRO124
ATHR125
ASER127
ASER147
AGLY148
ASER202
ALYS204
AHOH1061

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 483
ChainResidue
AGLU80
AGLN81
APHE82
AHOH1156
AHOH1161

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 484
ChainResidue
AASN95
ATHR98
AASN100
AHOH1200

site_idAC6
Number of Residues8
DetailsBINDING SITE FOR RESIDUE GOL A 486
ChainResidue
AGLN50
ACYS128
AALA129
ALYS230
AHOH1025
AHOH1073
AHOH1112
AHOH1125

site_idAC7
Number of Residues19
DetailsBINDING SITE FOR RESIDUE ANH A 487
ChainResidue
ALEU137
AASP189
AALA190
AGLN192
ASER195
AVAL200
ACYS201
ASER202
AGLY203
ATRP215
AGLY216
AGLY219
ACYS220
AGLY226
ASO4481
AHOH1001
AHOH1029
AHOH1121
AHOH1174

site_idAC8
Number of Residues9
DetailsBINDING SITE FOR RESIDUE GOL A 488
ChainResidue
ATYR39
AHIS40
AILE73
AASN74
AILE89
AVAL90
AHOH1092
AHOH1279
AHOH1281

Functional Information from PROSITE/UniProt
site_idPS00134
Number of Residues6
DetailsTRYPSIN_HIS Serine proteases, trypsin family, histidine active site. VSAAHC
ChainResidueDetails
AVAL53-CYS58

site_idPS00135
Number of Residues12
DetailsTRYPSIN_SER Serine proteases, trypsin family, serine active site. DAcqGDSGGPVV
ChainResidueDetails
AASP189-VAL200

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsACT_SITE: Charge relay system
ChainResidueDetails
AHIS57
AASP102
ASER195

site_idSWS_FT_FI2
Number of Residues7
DetailsBINDING:
ChainResidueDetails
AGLU70
AASN72
AVAL75
AGLU80
AASP189
AGLN192
ASER195

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PDB entries from 2024-07-17

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