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3UUD

Crystal structure of hERa-LBD (Y537S) in complex with estradiol

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EST A 600
ChainResidue
AHOH14
AMET343
ALEU346
AGLU353
AARG394
AHIS524
ALEU525

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL A 1
ChainResidue
AHOH577
AGLU323
ATRP393

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EST B 600
ChainResidue
BHOH4
BMET343
BLEU346
BGLU353
BARG394
BHIS524
BLEU525

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL B 1
ChainResidue
AHOH273
BHOH112
BASP351
BHOH572
BHOH575

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL B 553
ChainResidue
BHOH66
BGLU323
BTRP393
BGLY442
BHOH633

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO B 554
ChainResidue
BASN439
BGLN441
BALA493
BHOH626

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9338790","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"9600906","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1A52","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"1ERE","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Phosphotyrosine; by Tyr-kinases","evidences":[{"source":"PubMed","id":"7539106","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsLipidation: {"description":"S-palmitoyl cysteine","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 4"}
ChainResidueDetails

243083

PDB entries from 2025-10-15

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