3UUD
Crystal structure of hERa-LBD (Y537S) in complex with estradiol
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EST A 600 |
Chain | Residue |
A | HOH14 |
A | MET343 |
A | LEU346 |
A | GLU353 |
A | ARG394 |
A | HIS524 |
A | LEU525 |
site_id | AC2 |
Number of Residues | 3 |
Details | BINDING SITE FOR RESIDUE GOL A 1 |
Chain | Residue |
A | HOH577 |
A | GLU323 |
A | TRP393 |
site_id | AC3 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EST B 600 |
Chain | Residue |
B | HOH4 |
B | MET343 |
B | LEU346 |
B | GLU353 |
B | ARG394 |
B | HIS524 |
B | LEU525 |
site_id | AC4 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE GOL B 1 |
Chain | Residue |
A | HOH273 |
B | HOH112 |
B | ASP351 |
B | HOH572 |
B | HOH575 |
site_id | AC5 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE GOL B 553 |
Chain | Residue |
B | HOH66 |
B | GLU323 |
B | TRP393 |
B | GLY442 |
B | HOH633 |
site_id | AC6 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE EDO B 554 |
Chain | Residue |
B | ASN439 |
B | GLN441 |
B | ALA493 |
B | HOH626 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 6 |
Details | Binding site: {"evidences":[{"source":"PubMed","id":"9338790","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"9600906","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1A52","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"1ERE","evidenceCode":"ECO:0007744"}]} |
Chain | Residue | Details |
site_id | SWS_FT_FI2 |
Number of Residues | 2 |
Details | Modified residue: {"description":"Phosphotyrosine; by Tyr-kinases","evidences":[{"source":"PubMed","id":"7539106","evidenceCode":"ECO:0000269"}]} |
Chain | Residue | Details |
site_id | SWS_FT_FI3 |
Number of Residues | 2 |
Details | Lipidation: {"description":"S-palmitoyl cysteine","evidences":[{"evidenceCode":"ECO:0000250"}]} |
Chain | Residue | Details |
site_id | SWS_FT_FI4 |
Number of Residues | 8 |
Details | Motif: {"description":"LXXLL motif 4"} |
Chain | Residue | Details |