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3UPE

Bovine trypsin variant X(triplePhe227) in complex with small molecule inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004175molecular_functionendopeptidase activity
A0004252molecular_functionserine-type endopeptidase activity
A0005515molecular_functionprotein binding
A0005576cellular_componentextracellular region
A0005615cellular_componentextracellular space
A0006508biological_processproteolysis
A0007586biological_processdigestion
A0008236molecular_functionserine-type peptidase activity
A0046872molecular_functionmetal ion binding
A0097180cellular_componentserine protease inhibitor complex
A0097655molecular_functionserpin family protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA A 480
ChainResidue
AGLU70
AASN72
AVAL75
AGLU80
AHOH1001
AHOH1090

site_idAC2
Number of Residues20
DetailsBINDING SITE FOR RESIDUE 0CA A 481
ChainResidue
AASP189
AALA190
AGLN192
ASER195
ATRP215
AGLY216
ASER217
AGLY219
ACYS220
AGLY226
AHOH1011
AHOH1024
AHOH1118
AHOH1121
AHOH1126
AHOH1151
AHOH1202
AGLU97
ATYR99
APHE174

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 483
ChainResidue
ATHR177
ASER178
ALYS188
AHOH1139

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 484
ChainResidue
AASN95
AASN100
AHOH1124
AHOH1226
AHOH1289

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 485
ChainResidue
AGLU80
APHE82
AHOH1164
AHOH1188
AHOH1229

Functional Information from PROSITE/UniProt
site_idPS00134
Number of Residues6
DetailsTRYPSIN_HIS Serine proteases, trypsin family, histidine active site. VSAAHC
ChainResidueDetails
AVAL53-CYS58

site_idPS00135
Number of Residues12
DetailsTRYPSIN_SER Serine proteases, trypsin family, serine active site. DAcqGDSGGPVV
ChainResidueDetails
AASP189-VAL200

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsACT_SITE: Charge relay system
ChainResidueDetails
AHIS57
AASP102
ASER195

site_idSWS_FT_FI2
Number of Residues7
DetailsBINDING:
ChainResidueDetails
AGLU70
AASN72
AVAL75
AGLU80
AASP189
AGLN192
ASER195

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PDB entries from 2024-07-31

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