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3U9Y

Crystal structure of human tankyrase 2 catalytic domain in complex with olaparib

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1163
ChainResidue
ALYS1067
AHOH99
AHOH100
AARG977
AHIS979
AARG980

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 2
ChainResidue
AASN990
AARG991
AGLU1161

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 1164
ChainResidue
AHOH62
AGLU978
AHIS979
AILE988
APHE989

site_idAC5
Number of Residues16
DetailsBINDING SITE FOR RESIDUE 09L A 1165
ChainResidue
AHOH48
AHIS1031
AGLY1032
AILE1039
AASP1045
AHIS1048
AALA1049
ATYR1050
AGLY1058
AILE1059
ATYR1060
AALA1062
ASER1068
ATYR1071
AILE1075
AGLU1138

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092

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PDB entries from 2024-07-10

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