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3T3U

Calcium-Dependent Protein Kinase 1 from Toxoplasma gondii (TgCDPK1) in complex with Bumped Kinase Inhibitor, RM-1-130

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0004674molecular_functionprotein serine/threonine kinase activity
A0005509molecular_functioncalcium ion binding
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
A0016020cellular_componentmembrane
A0046872molecular_functionmetal ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE BK6 A 701
ChainResidue
AVAL65
AGLU178
ALEU181
AASP195
AEDO712
AHOH825
AALA78
ALYS80
AMET112
ALEU114
ALEU126
AGLU129
ATYR131
AGLU135

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE DMS A 711
ChainResidue
ATYR267
AARG286
AGLY420
ATYR421

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 712
ChainResidue
AMET112
APHE196
ABK6701
AHOH809

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 713
ChainResidue
AGLY225
ATHR226
ATYR227
AGLU444
AARG448

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 714
ChainResidue
ASER160
ATHR163
ATYR164
ALYS167

Functional Information from PROSITE/UniProt
site_idPS00018
Number of Residues13
DetailsEF_HAND_1 EF-hand calcium-binding domain. DKNGDGQLDraEL
ChainResidueDetails
AASP368-LEU380
AASP415-PHE427
AASP451-LEU463
AASP485-PHE497

site_idPS00107
Number of Residues24
DetailsPROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. LGKGSFGEVIlCkdkitgqe..........CAVK
ChainResidueDetails
ALEU57-LYS80

site_idPS00108
Number of Residues13
DetailsPROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. IvHrDLKpeNLLL
ChainResidueDetails
AILE170-LEU182

222624

PDB entries from 2024-07-17

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