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3SU2

Crystal structure of NS3/4A protease variant A156T in complex with danoprevir

Functional Information from GO Data
ChainGOidnamespacecontents
A0006508biological_processproteolysis
A0008236molecular_functionserine-type peptidase activity
A0019087biological_processtransformation of host cell by virus
Functional Information from PDB Data
site_idAC1
Number of Residues21
DetailsBINDING SITE FOR RESIDUE TSV A 100
ChainResidue
AHOH47
AVAL1078
AASP1079
AASP1081
ALEU1135
ALYS1136
AGLY1137
ASER1138
AALA1139
APHE1154
AARG1155
AHOH69
ATHR1156
AALA1157
AHOH133
AHOH140
AHOH147
AGLN1041
APHE1043
AHIS1057
AGLY1058

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 1
ChainResidue
AHOH13
AHOH34
AHOH39
ATYR1006
AGLN1008
ATYR1056
AHOH1186

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 2
ChainResidue
AHOH50
AHOH72
AHOH83
AHOH108
AARG1109
AHIS1110

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1183
ChainResidue
ACYS1097
ACYS1099
ACYS1145
AHIS1149

219869

PDB entries from 2024-05-15

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