Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

3SKA

I. Novel HCV NS5B Polymerase Inhibitors: Discovery of Indole 2- Carboxylic Acids with C3-Heterocycles

Functional Information from GO Data
ChainGOidnamespacecontents
A0003723molecular_functionRNA binding
A0003968molecular_functionRNA-dependent RNA polymerase activity
A0039694biological_processviral RNA genome replication
B0003723molecular_functionRNA binding
B0003968molecular_functionRNA-dependent RNA polymerase activity
B0039694biological_processviral RNA genome replication
Functional Information from PDB Data
site_idAC1
Number of Residues9
DetailsBINDING SITE FOR RESIDUE PO4 A 577
ChainResidue
APRO265
AARG505
AVAL530
AARG531
ATHR532
AHOH662
AHOH772
AHOH980
AHOH1058

site_idAC2
Number of Residues17
DetailsBINDING SITE FOR RESIDUE 053 A 578
ChainResidue
APRO197
AASN316
ACYS366
ASER367
ASER368
ALEU384
AGLY410
AASN411
AMET414
ATYR415
AGLN446
AILE447
ATYR448
AHOH825
AHOH1072
AHOH4014
AHOH4025

site_idAC3
Number of Residues14
DetailsBINDING SITE FOR RESIDUE 053 B 577
ChainResidue
BPRO197
BASN316
BCYS366
BSER368
BLEU384
BGLY410
BASN411
BMET414
BTYR415
BGLN446
BILE447
BTYR448
BHOH691
BHOH832

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P26663
ChainResidueDetails
AASP220
AASP318
AASP319
BASP220
BASP318
BASP319

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: Phosphoserine; by host => ECO:0000250|UniProtKB:P26662
ChainResidueDetails
ASER29
ASER42
BSER29
BSER42

224931

PDB entries from 2024-09-11

PDB statisticsPDBj update infoContact PDBjnumon