3S91
Crystal Structure of the first bromodomain of human BRD3 in complex with the inhibitor JQ1
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 10 |
Details | BINDING SITE FOR RESIDUE JQ1 A 1 |
Chain | Residue |
A | HOH5 |
A | MET125 |
A | TRP57 |
A | TRP57 |
A | PRO58 |
A | VAL63 |
A | LEU68 |
A | LEU70 |
A | ASN116 |
A | ILE122 |
site_id | AC2 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE IPA A 145 |
Chain | Residue |
A | TYR94 |
A | GLU100 |
A | HOH198 |
A | HOH198 |
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 60 |
Details | BROMODOMAIN_1 Bromodomain signature. AwpFyqpvDaiklnlpDYHkiIknpMdmgtIkkrlenny..Ywsasecmqdfnt.MftNCyiY |
Chain | Residue | Details |
A | ALA56-TYR115 |