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3S3N

Crystal structure of the Prototype Foamy Virus (PFV) S217H mutant intasome in complex with magnesium and Dolutegravir (S/GSK1349572)

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 393
ChainResidue
AHIS62
AHIS66
ACYS96
ACYS99

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 394
ChainResidue
AHIS338
ALYS339
AHOH427

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL A 801
ChainResidue
ASER164
ASER162
ATHR163

site_idAC4
Number of Residues2
DetailsBINDING SITE FOR RESIDUE GOL A 802
ChainResidue
AGLN137
ALYS241

site_idAC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE GOL A 803
ChainResidue
AGLN296
BASP273

site_idAC6
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 805
ChainResidue
AGLN60
ALEU79
ATYR80
APRO277
APHE278

site_idAC7
Number of Residues1
DetailsBINDING SITE FOR RESIDUE NH4 A 395
ChainResidue
AASP116

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MG A 396
ChainResidue
AASP128
AASP185
ADLU398
AHOH400
AHOH527

site_idAC9
Number of Residues4
DetailsBINDING SITE FOR RESIDUE MG A 397
ChainResidue
AASP128
AGLU221
ADLU398
AHOH528

site_idBC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE DLU A 398
ChainResidue
AASP128
AASP185
APRO214
AGLN215
AGLU221
AMG396
AMG397
AHOH400
AHOH521
AHOH527
CDG4
DDC16
DDA17

site_idBC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 399
ChainResidue
AARG114
ATYR303
APRO305
AHOH529
CDC6

site_idBC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 393
ChainResidue
BLYS219
BARG222
BSER258
BPRO259
BVAL260

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues156
DetailsDomain: {"description":"Integrase catalytic","evidences":[{"source":"PROSITE-ProRule","id":"PRU00457","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsBinding site: {"evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

245663

PDB entries from 2025-12-03

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