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3RXW

KPC-2 carbapenemase in complex with PSR3-226

Functional Information from GO Data
ChainGOidnamespacecontents
A0008800molecular_functionbeta-lactamase activity
A0016787molecular_functionhydrolase activity
A0017001biological_processantibiotic catabolic process
A0030655biological_processbeta-lactam antibiotic catabolic process
A0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues17
DetailsBINDING SITE FOR RESIDUE SR3 A 1
ChainResidue
ASER69
AGLY235
ATHR236
APRO251
ATHR252
ACIT290
AHOH313
AHOH316
AHOH579
APRO103
ATRP104
AASN131
AGLU165
ALEU166
AASN169
AASP227
ATRP228

site_idAC2
Number of Residues14
DetailsBINDING SITE FOR RESIDUE CIT A 290
ChainResidue
ASR31
ASER69
ATRP104
ASER129
ATHR215
AARG219
ALYS233
ATHR234
AGLY235
ATHR236
AARG254
AHOH298
AHOH312
AHOH318

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: Acyl-ester intermediate => ECO:0000250
ChainResidueDetails
ASER69

site_idSWS_FT_FI2
Number of Residues1
DetailsACT_SITE: Proton acceptor => ECO:0000250
ChainResidueDetails
AGLU167

site_idSWS_FT_FI3
Number of Residues1
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
ALYS233

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PDB entries from 2024-07-10

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