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3R0Y

Crystal Structures of Multidrug-resistant HIV-1 Protease in Complex with Mechanism-Based Aspartyl Protease Inhibitors

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues20
DetailsBINDING SITE FOR RESIDUE RSZ A 301
ChainResidue
AASN25
AHOH165
AHOH190
AHOH195
BASN25
BGLY27
BGLY48
BTHR80
BPRO81
BTHR82
BHOH102
AGLY27
BHOH166
AILE50
AGLN61
ATHR80
APRO81
ATHR82
AVAL84
AHOH110

231564

PDB entries from 2025-02-19

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