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3Q81

Imipenem acylated BlaR1 sensor domain from Staphylococcus aureus

Functional Information from GO Data
ChainGOidnamespacecontents
A0008658molecular_functionpenicillin binding
B0008658molecular_functionpenicillin binding
Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE IM2 A 254
ChainResidue
AASN58
AGLY198
ATHR199
ASER59
APHE91
AALA93
AASN106
ASER107
AASN109
ALYS196
ATHR197

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GOL A 1
ChainResidue
ALYS87
ATYR89
BLYS87
BTYR89

site_idAC3
Number of Residues12
DetailsBINDING SITE FOR RESIDUE IM2 B 254
ChainResidue
BASN58
BSER59
BPHE91
BALA93
BTRP94
BASN106
BSER107
BASN109
BLYS196
BTHR197
BGLY198
BTHR199

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsActive site: {"description":"Acyl-ester intermediate","evidences":[{"source":"PubMed","id":"15506754","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"21775440","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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