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3Q2F

Crystal Structure of the bromodomain of human BAZ2B in complex with a triazolo ligand

Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE OAM A 1
ChainResidue
AEDO3
AASN1944
AHOH12
AHOH64
APRO1862
ATRP1887
APRO1888
AVAL1893
AVAL1898
APRO1899

site_idAC2
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 1973
ChainResidue
AGLU1881
AARG1915

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2
ChainResidue
ALEU1872
AMET1875
AGLU1879
ALYS1964
ATHR1968

site_idAC4
Number of Residues8
DetailsBINDING SITE FOR RESIDUE EDO A 3
ChainResidue
AOAM1
AHOH33
AHOH110
ATRP1887
APRO1888
ALEU1890
ALEU1891
APRO1892

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFllpvNlklvp..GYKkvIkkpMdfstIreklssgq..Ypnletfaldvrl.VfdNCetF
ChainResidueDetails
AALA1886-PHE1943

225946

PDB entries from 2024-10-09

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