Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

3PYH

Bovine trypsin variant X(tripleGlu217Ile227) in complex with small molecule inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004175molecular_functionendopeptidase activity
A0004252molecular_functionserine-type endopeptidase activity
A0005515molecular_functionprotein binding
A0005576cellular_componentextracellular region
A0005615cellular_componentextracellular space
A0006508biological_processproteolysis
A0007586biological_processdigestion
A0008236molecular_functionserine-type peptidase activity
A0046872molecular_functionmetal ion binding
A0097180cellular_componentserine protease inhibitor complex
A0097655molecular_functionserpin family protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA A 480
ChainResidue
AGLU70
AASN72
AVAL75
AGLU80
AHOH1009
AHOH1013

site_idAC2
Number of Residues23
DetailsBINDING SITE FOR RESIDUE 3YH A 481
ChainResidue
APHE174
ATYR184
ALEU185
AGLU186
ALYS188
AASP189
AALA190
AGLN192
ASER195
ATRP215
AGLY216
AGLY219
AGLY226
AHOH1004
AHOH1042
AHOH1059
AHOH1094
AHOH1101
AHOH1124
AHOH1190
AGLU97
ATHR98
ATYR99

site_idAC3
Number of Residues9
DetailsBINDING SITE FOR RESIDUE SO4 A 482
ChainResidue
AHIS57
AGLN135
AGLN192
AGLY193
ASER195
AHOH1114
AHOH1120
AHOH1132
AHOH1260

site_idAC4
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A 483
ChainResidue
AASP153
AHOH1246

Functional Information from PROSITE/UniProt
site_idPS00134
Number of Residues6
DetailsTRYPSIN_HIS Serine proteases, trypsin family, histidine active site. VSAAHC
ChainResidueDetails
AVAL53-CYS58

site_idPS00135
Number of Residues12
DetailsTRYPSIN_SER Serine proteases, trypsin family, serine active site. DAcqGDSGGPVV
ChainResidueDetails
AASP189-VAL200

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsACT_SITE: Charge relay system
ChainResidueDetails
AHIS57
AASP102
ASER195

site_idSWS_FT_FI2
Number of Residues7
DetailsBINDING:
ChainResidueDetails
AGLU70
AASN72
AVAL75
AGLU80
AASP189
AGLN192
ASER195

222624

PDB entries from 2024-07-17

PDB statisticsPDBj update infoContact PDBjnumon