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3PO9

Crystal structure of PPARgamma ligand binding domain in complex with tripropyltin

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues20
DetailsBINDING SITE FOR RESIDUE XPT A 1
ChainResidue
AHOH152
ALEU353
APHE360
APHE363
AMET364
ALYS367
AHIS449
ALEU453
ATYR473
AHOH508
AHOH509
APHE282
AHOH528
ACYS285
AARG288
ATYR327
ALEU330
AVAL339
AILE341
AMET348

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE XPT B 1
ChainResidue
BPGO4
BCYS285
BTYR327
BMET364
BPGO478

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE PGO B 478
ChainResidue
BXPT1
BPGO4
BCYS285
BARG288
BHOH481

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE PGO B 2
ChainResidue
BARG397
BPRO398
BARG443
BHOH495

site_idAC5
Number of Residues1
DetailsBINDING SITE FOR RESIDUE PGO B 3
ChainResidue
BTYR320

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PGO B 4
ChainResidue
BXPT1
BHOH169
BCYS285
BARG288
BSER289
BPGO478

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues16
DetailsMotif: {"description":"9aaTAD","evidences":[{"source":"PubMed","id":"30468856","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues12
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9744270","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2PRG","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"36737649","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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