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3PAE

Crystal structure of the K84D mutant of OXA-24/40 in complex with doripenem

Functional Information from GO Data
ChainGOidnamespacecontents
A0008658molecular_functionpenicillin binding
A0008800molecular_functionbeta-lactamase activity
A0016787molecular_functionhydrolase activity
A0071555biological_processcell wall organization
B0008658molecular_functionpenicillin binding
B0008800molecular_functionbeta-lactamase activity
B0016787molecular_functionhydrolase activity
B0071555biological_processcell wall organization
Functional Information from PDB Data
site_idAC1
Number of Residues18
DetailsBINDING SITE FOR RESIDUE 4J6 A 300
ChainResidue
AHOH8
ATRP221
AMET223
AGLY258
ASER259
AARG261
AHOH284
AHOH390
AHOH392
AHOH406
AALA80
ASER81
ATRP115
ALEU127
ASER128
ALEU168
ASER219
AGLY220

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1
ChainResidue
AGLY141
ALEU142
AGLU143
AHOH288
AHOH364

site_idAC3
Number of Residues18
DetailsBINDING SITE FOR RESIDUE 4J6 B 300
ChainResidue
BALA80
BSER81
BTRP115
BLEU127
BSER128
BVAL130
BLEU168
BSER219
BGLY220
BTRP221
BMET223
BGLY258
BSER259
BARG261
BHOH314
BHOH351
BHOH355
BHOH401

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 2
ChainResidue
AHOH356
BGLY141
BLEU142
BGLU143

site_idAC5
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 3
ChainResidue
BGLU76
BTYR77
BVAL78
BVAL225
BPRO227
BVAL229
BHOH402

221051

PDB entries from 2024-06-12

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