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3P8H

Crystal structure of L3MBTL1 (MBT repeat) in complex with a nicotinamide antagonist

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
C0005634cellular_componentnucleus
C0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE P8H A 600
ChainResidue
AASP355
BGLN406
AASN358
ASER360
ALEU361
ACYS363
APHE379
ATRP382
ATYR386
BTRP402

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 610
ChainResidue
ATYR275
ASER276
AHIS279
ALYS307

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 620
ChainResidue
APRO221
AVAL222
ASER223
CSER487
CTYR490

site_idAC4
Number of Residues1
DetailsBINDING SITE FOR RESIDUE GOL A 621
ChainResidue
AASP248

site_idAC5
Number of Residues7
DetailsBINDING SITE FOR RESIDUE P8H B 600
ChainResidue
BASP355
BASN358
BSER360
BLEU361
BCYS363
BTRP382
BTYR386

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 610
ChainResidue
BTYR275
BSER276
BHIS279
BLYS307

site_idAC7
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 C 610
ChainResidue
CTYR275
CSER276
CHIS279
CLYS307

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues300
DetailsRepeat: {"description":"MBT 1"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues297
DetailsRepeat: {"description":"MBT 2"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues285
DetailsRepeat: {"description":"MBT 3"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues21
DetailsRegion: {"description":"Interaction with monomethylated and dimethylated peptides"}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues3
DetailsSite: {"description":"Mediates recognition of monomethylated and dimethylated peptides"}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues3
DetailsSite: {"description":"Positioned at the entrance of MBT 2 and is required for recognition of monomethylated and dimethylated peptides"}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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