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3KI5

Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-M

Functional Information from GO Data
ChainGOidnamespacecontents
A0047286molecular_functionNAD+-diphthamide ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE G9M A 1
ChainResidue
AHOH135
AGLU581
AHOH187
ATYR459
AHIS460
AGLY461
AASN485
ATYR493
AALA501
ATYR504

site_idAC2
Number of Residues12
DetailsBINDING SITE FOR RESIDUE G9M A 635
ChainResidue
AHOH124
AHOH148
AHOH163
AHOH231
AALA448
ALEU449
ATYR454
AGLU513
ATYR514
AASN550
AGLU553
AVAL593

Functional Information from PROSITE/UniProt
site_idPS00014
Number of Residues4
DetailsER_TARGET Endoplasmic reticulum targeting sequence. KDEL
ChainResidueDetails
ALYS630-LEU633

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: ACT_SITE => ECO:0000305
ChainResidueDetails
AGLU581

226262

PDB entries from 2024-10-16

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