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3KI4

Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-P

Functional Information from GO Data
ChainGOidnamespacecontents
A0047286molecular_functionNAD+-diphthamide ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE G9P A 1
ChainResidue
AHOH23
AHOH178
AHIS460
AGLY461
ATYR493
AALA501
ATYR504
AGLU581

site_idAC2
Number of Residues12
DetailsBINDING SITE FOR RESIDUE GOL A 3968
ChainResidue
AHOH11
AHOH13
AHOH242
AHOH250
AVAL471
AASN472
AARG473
AGLU549
AASN550
AALA576
AVAL593
AHOH4

site_idAC3
Number of Residues8
DetailsBINDING SITE FOR RESIDUE GOL A 635
ChainResidue
AHOH59
AHOH155
AHIS446
APHE456
ASER619
AILE620
ASER621
ATHR622

Functional Information from PROSITE/UniProt
site_idPS00014
Number of Residues4
DetailsER_TARGET Endoplasmic reticulum targeting sequence. KDEL
ChainResidueDetails
ALYS630-LEU633

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: ACT_SITE => ECO:0000305
ChainResidueDetails
AGLU581

222415

PDB entries from 2024-07-10

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