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3IPQ

X-ray structure of GW3965 synthetic agonist bound to the LXR-alpha

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006629biological_processlipid metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues19
DetailsBINDING SITE FOR RESIDUE 965 A 801
ChainResidue
AHOH66
APHE315
ALEU316
APHE326
APHE335
AILE339
AHIS421
AGLN424
ALEU428
ALEU435
ATRP443
APHE257
ALEU260
AALA261
ASER264
AMET298
ALEU299
ATHR302
AARG305

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 B 802
ChainResidue
AARG283
AARG283
BHOH76
BHOH76
BHIS690
BHIS690
BGLN694
BGLN694

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 4"}
ChainResidueDetails

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PDB entries from 2025-12-17

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