3H7W
Crystal structure of the high affinity heterodimer of HIF2 alpha and ARNT C-terminal PAS domains with the artificial ligand THS017
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 14 |
Details | BINDING SITE FOR RESIDUE 018 A 1 |
Chain | Residue |
A | HIS248 |
A | TYR307 |
A | MET309 |
A | THR321 |
A | CYS339 |
A | ASN341 |
A | MET252 |
A | ALA277 |
A | TYR281 |
A | MET289 |
A | SER292 |
A | HIS293 |
A | VAL302 |
A | SER304 |