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3H7W

Crystal structure of the high affinity heterodimer of HIF2 alpha and ARNT C-terminal PAS domains with the artificial ligand THS017

Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE 018 A 1
ChainResidue
AHIS248
ATYR307
AMET309
ATHR321
ACYS339
AASN341
AMET252
AALA277
ATYR281
AMET289
ASER292
AHIS293
AVAL302
ASER304

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues43
DetailsDomain: {"description":"PAC"}
ChainResidueDetails

246905

PDB entries from 2025-12-31

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