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3GYN

Crystal structure of HCV NS5B polymerase with a novel monocyclic dihydropyridinone inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003723molecular_functionRNA binding
A0003968molecular_functionRNA-dependent RNA polymerase activity
A0039694biological_processviral RNA genome replication
B0003723molecular_functionRNA binding
B0003968molecular_functionRNA-dependent RNA polymerase activity
B0039694biological_processviral RNA genome replication
Functional Information from PDB Data
site_idAC1
Number of Residues20
DetailsBINDING SITE FOR RESIDUE B42 A 579
ChainResidue
APHE193
AGLY410
AASN411
AMET414
ATYR415
AGLN446
AILE447
ATYR448
AGLY449
ASER556
AHOH582
ASER288
AHOH623
AASN291
AASN316
AGLY317
AASP318
ACYS366
ALEU384
AARG386

site_idAC2
Number of Residues19
DetailsBINDING SITE FOR RESIDUE B42 B 579
ChainResidue
BPHE193
BSER288
BASN291
BASN316
BGLY317
BASP318
BCYS366
BLEU384
BARG386
BGLY410
BASN411
BMET414
BTYR415
BGLN446
BTYR448
BGLY449
BSER556
BHOH606
BHOH610

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000305|PubMed:10557268, ECO:0000305|PubMed:11884572
ChainResidueDetails
AASP220
AASP318
AASP319
BASP220
BASP318
BASP319

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: Phosphoserine; by host => ECO:0000250|UniProtKB:P26662
ChainResidueDetails
ASER29
ASER42
BSER29
BSER42

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PDB entries from 2024-04-24

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