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3G30

CTX-M-9 class A beta-lactamase complexed with compound 3 (G30)

Functional Information from GO Data
ChainGOidnamespacecontents
A0008800molecular_functionbeta-lactamase activity
A0016787molecular_functionhydrolase activity
A0017001biological_processantibiotic catabolic process
A0030655biological_processbeta-lactam antibiotic catabolic process
A0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE G30 A 1
ChainResidue
ASER70
AHOH311
AHOH347
AASN104
ASER130
AASN132
AASN170
ASER237
AGLY238
AASP240
AHOH309

site_idAC2
Number of Residues12
DetailsBINDING SITE FOR RESIDUE G30 A 2
ChainResidue
AG303
AGLN83
ALEU142
AGLY146
ATHR149
AALA150
AALA150
AARG153
AHOH303
AHOH356
AHOH368
AHOH414

site_idAC3
Number of Residues10
DetailsBINDING SITE FOR RESIDUE G30 A 3
ChainResidue
AG302
AALA79
ALYS82
AGLN83
AALA150
APHE151
AARG153
AALA154
AHOH367
AHOH420

Functional Information from PROSITE/UniProt
site_idPS00146
Number of Residues16
DetailsBETA_LACTAMASE_A Beta-lactamase class-A active site. FpMCSTsKvmaAAAVL
ChainResidueDetails
APHE66-LEU81

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PDB entries from 2024-06-12

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