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3DY6

PPARdelta complexed with an anthranilic acid partial agonist

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE DY6 A 478
ChainResidue
AARG284
AHIS449
ATYR473
ACYS285
ATHR288
ATHR289
APHE327
ALEU330
ALEU339
AILE364
ALYS367

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE DY6 B 1
ChainResidue
BTRP264
BCYS285
BTHR288
BTHR289
BPHE327
BLEU330
BLEU339
BILE364
BHIS449
BTYR473

219140

PDB entries from 2024-05-01

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