3DY6
PPARdelta complexed with an anthranilic acid partial agonist
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0003677 | molecular_function | DNA binding |
A | 0004879 | molecular_function | nuclear receptor activity |
A | 0005634 | cellular_component | nucleus |
A | 0006355 | biological_process | regulation of DNA-templated transcription |
B | 0003677 | molecular_function | DNA binding |
B | 0004879 | molecular_function | nuclear receptor activity |
B | 0005634 | cellular_component | nucleus |
B | 0006355 | biological_process | regulation of DNA-templated transcription |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 11 |
Details | BINDING SITE FOR RESIDUE DY6 A 478 |
Chain | Residue |
A | ARG284 |
A | HIS449 |
A | TYR473 |
A | CYS285 |
A | THR288 |
A | THR289 |
A | PHE327 |
A | LEU330 |
A | LEU339 |
A | ILE364 |
A | LYS367 |
site_id | AC2 |
Number of Residues | 10 |
Details | BINDING SITE FOR RESIDUE DY6 B 1 |
Chain | Residue |
B | TRP264 |
B | CYS285 |
B | THR288 |
B | THR289 |
B | PHE327 |
B | LEU330 |
B | LEU339 |
B | ILE364 |
B | HIS449 |
B | TYR473 |