Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

3AO1

Fragment-based approach to the design of ligands targeting a novel site in HIV-1 integrase

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD A 1003
ChainResidue
ACYS65
AHIS67
AGLU92
ACD1004
BASP131
BHOH223

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE CD A 1004
ChainResidue
AGLU92
AASP116
ACD1003
BASP131
AHOH4
AHOH30
ACYS65

site_idAC3
Number of Residues9
DetailsBINDING SITE FOR RESIDUE SO4 A 1
ChainResidue
AHOH11
AGLU69
ALYS71
AARG166
AGLU170
AHIS171
ALEU172
AARG187
AHOH221

site_idAC4
Number of Residues9
DetailsBINDING SITE FOR RESIDUE BZX A 213
ChainResidue
AHOH31
ATYR83
AASN184
AHIS185
AGLY197
AVAL201
BGLY106
BARG107
BPRO109

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE BZX A 214
ChainResidue
AHOH9
AGLY70
AHIS185
BPRO109

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD B 1001
ChainResidue
BHOH3
BCYS65
BGLU92
BASP116
BHOH213
BCD1002

site_idAC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CD B 1002
ChainResidue
BCYS65
BHIS67
BGLU92
BHOH224
BCD1001

site_idAC8
Number of Residues12
DetailsBINDING SITE FOR RESIDUE BZX B 1
ChainResidue
AGLY106
AARG107
ATRP108
APRO109
BHOH22
BHOH36
BTYR83
BASN184
BHIS185
BGLY197
BGLU198
BHOH225

219140

PDB entries from 2024-05-01

PDB statisticsPDBj update infoContact PDBjnumon