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36JD

Crystal structure of Yck2 from Candida albicans in complex with kinase inhibitor MN-III-28: N-(4-(6-cyano-2-(4-fluorophenyl)pyrazolo[1,5-a]pyridin-3-yl)pyridin-2-yl)acetamide

This is a non-PDB format compatible entry.
Functional Information from PROSITE/UniProt
site_idPS00107
Number of Residues24
DetailsPROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGEGSFGVIFeGtniingvp..........VAIK
ChainResidueDetails
AILE50-LYS73

site_idPS00108
Number of Residues13
DetailsPROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. LiYrDIKpdNFLI
ChainResidueDetails
ALEU159-ILE171

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues267
DetailsDomain: {"description":"Protein kinase","evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsActive site: {"description":"Proton acceptor","evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues9
DetailsBinding site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

259351

PDB entries from 2026-09-09

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