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2YUU

Solution structure of the first Phorbol esters/diacylglycerol binding domain of human Protein kinase C, delta

Functional Information from GO Data
ChainGOidnamespacecontents
A0004674molecular_functionprotein serine/threonine kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE ZN A 201
ChainResidue
AHIS18
AGLU19
APHE20

site_idAC2
Number of Residues2
DetailsBINDING SITE FOR RESIDUE ZN A 401
ChainResidue
ACYS31
ACYS34

Functional Information from PROSITE/UniProt
site_idPS00479
Number of Residues50
DetailsZF_DAG_PE_1 Zinc finger phorbol-ester/DAG-type signature. HeFiatffgqptf.CsvCkdfVwglnkqgyk.CrqCnaaiHkkCidkiigr..C
ChainResidueDetails
AHIS18-CYS67

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues50
DetailsZN_FING: Phorbol-ester/DAG-type 1 => ECO:0000255|PROSITE-ProRule:PRU00226
ChainResidueDetails
AASN17-CYS67

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0000269|PubMed:15774464
ChainResidueDetails
ATYR14

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: Phosphothreonine => ECO:0007744|PubMed:19369195
ChainResidueDetails
ATHR77

218853

PDB entries from 2024-04-24

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