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2XGM

Substrate and product analogues as human O-GlcNAc transferase inhibitors.

Functional Information from GO Data
ChainGOidnamespacecontents
A0016740molecular_functiontransferase activity
A0016757molecular_functionglycosyltransferase activity
A0046872molecular_functionmetal ion binding
A0097363molecular_functionprotein O-acetylglucosaminyltransferase activity
B0016740molecular_functiontransferase activity
B0016757molecular_functionglycosyltransferase activity
B0046872molecular_functionmetal ion binding
B0097363molecular_functionprotein O-acetylglucosaminyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE LXN A 1569
ChainResidue
ALEU412
ALEU442
AHIS444
ATYR447

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE LXN B 1569
ChainResidue
BLEU412
BLEU442
BHIS444
BTYR447

246704

PDB entries from 2025-12-24

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