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2V11

Crystal Structure of Renin with Inhibitor 6

Functional Information from GO Data
ChainGOidnamespacecontents
C0004190molecular_functionaspartic-type endopeptidase activity
C0006508biological_processproteolysis
O0004190molecular_functionaspartic-type endopeptidase activity
O0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues17
DetailsBINDING SITE FOR RESIDUE C80 C1341
ChainResidue
CTHR18
CALA122
CPHE124
CGLN135
CASP226
CTHR227
CGLY228
CALA229
CSER230
CTYR20
CVAL36
CASP38
CSER41
CSER42
CTYR83
CSER84
CTHR85

site_idAC2
Number of Residues22
DetailsBINDING SITE FOR RESIDUE C80 O1341
ChainResidue
OTHR18
OGLN19
OTYR20
OVAL36
OASP38
OGLY40
OSER41
OARG82
OTYR83
OSER84
OTHR85
OPRO118
OLEU121
OALA122
OGLN135
OILE137
OASP226
OTHR227
OGLY228
OALA229
OSER230
OILE305

Functional Information from PROSITE/UniProt
site_idPS00141
Number of Residues12
DetailsASP_PROTEASE Eukaryotic and viral aspartyl proteases active site. VVFDTGSSNVWV
ChainResidueDetails
CVAL35-VAL46
CALA223-GLY234

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsACT_SITE: ACT_SITE => ECO:0000269|PubMed:20927107
ChainResidueDetails
CASP38
CASP226
OASP38
OASP226

site_idSWS_FT_FI2
Number of Residues4
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:2493678
ChainResidueDetails
CASN5
CASN75
OASN5
OASN75

Catalytic Information from CSA
site_idCSA1
Number of Residues4
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
CASP38
CASP226
CTHR39
CTHR227

site_idCSA10
Number of Residues2
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
OASP226
OTHR32

site_idCSA2
Number of Residues4
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
OASP38
OASP226
OTHR39
OTHR227

site_idCSA3
Number of Residues3
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
CASP38
CASP226
CSER41

site_idCSA4
Number of Residues3
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
OASP38
OASP226
OSER41

site_idCSA5
Number of Residues4
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
CASP38
CASP226
CTYR83
CSER41

site_idCSA6
Number of Residues4
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
OASP38
OASP226
OTYR83
OSER41

site_idCSA7
Number of Residues1
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
CASP38

site_idCSA8
Number of Residues1
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
OASP38

site_idCSA9
Number of Residues2
DetailsAnnotated By Reference To The Literature 1avf
ChainResidueDetails
CASP226
CTHR32

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数据于2024-09-18公开中

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